Cerdulatinib hydrochloride

CAS No. 1369761-01-2

Cerdulatinib hydrochloride ( —— )

Catalog No. M17977 CAS No. 1369761-01-2

Cerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 78 Get Quote
10MG 105 Get Quote
25MG 201 Get Quote
50MG 354 Get Quote
100MG 527 Get Quote
500MG 1143 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Cerdulatinib hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Cerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively.
  • Description
    Cerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively. Also inhibits 19 other tested kinases with IC50 less than 200 nM.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    c-Fms; MST1; ARK5; MLK1; Tyk2
  • Research Area
    Cancer|Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    1369761-01-2
  • Formula Weight
    482
  • Molecular Formula
    C20H28ClN7O3S
  • Purity
    98%
  • Solubility
    ——
  • SMILES
    Cl.CCS(=O)(=O)N1CCN(CC1)C1=CC=C(NC2=NC(NC3CC3)=C(C=N2)C(N)=O)C=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Coffey G, J Pharmacol Exp Ther. 2014, 351(3), 538-548.
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