Cerdulatinib hydrochloride
CAS No. 1369761-01-2
Cerdulatinib hydrochloride ( —— )
Catalog No. M17977 CAS No. 1369761-01-2
Cerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 78 | Get Quote |
|
10MG | 105 | Get Quote |
|
25MG | 201 | Get Quote |
|
50MG | 354 | Get Quote |
|
100MG | 527 | Get Quote |
|
500MG | 1143 | Get Quote |
|
1G | Get Quote | Get Quote |
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Biological Information
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Product NameCerdulatinib hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionCerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively.
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DescriptionCerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively. Also inhibits 19 other tested kinases with IC50 less than 200 nM.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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Recptorc-Fms; MST1; ARK5; MLK1; Tyk2
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Research AreaCancer|Inflammation/Immunology
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Indication——
Chemical Information
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CAS Number1369761-01-2
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Formula Weight482
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Molecular FormulaC20H28ClN7O3S
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Purity98%
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Solubility——
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SMILESCl.CCS(=O)(=O)N1CCN(CC1)C1=CC=C(NC2=NC(NC3CC3)=C(C=N2)C(N)=O)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Coffey G, J Pharmacol Exp Ther. 2014, 351(3), 538-548.
molnova catalog
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